Metheptazine

Metheptazine is an opioid analgesic from the phenazepane family. It was developed by American Home Products in the 1950s.[1]

Metheptazine
Clinical data
Other namesMetheptazine
ATC code
  • none
Identifiers
  • methyl 1,2-dimethyl-4-phenylazepane-4-carboxylate
CAS Number
PubChem CID
ChemSpider
UNII
ChEMBL
Chemical and physical data
FormulaC16H23NO2
Molar mass261.365 g·mol−1
3D model (JSmol)
  • O=C(OC)C2(c1ccccc1)CC(N(C)CCC2)C
  • InChI=1S/C16H23NO2/c1-13-12-16(15(18)19-3,10-7-11-17(13)2)14-8-5-4-6-9-14/h4-6,8-9,13H,7,10-12H2,1-3H3 Y
  • Key:RAAFYFKWMRWOIT-UHFFFAOYSA-N Y
 NY (what is this?)  (verify)

Metheptazine produces similar effects to other opioids, including analgesia, sedation, dizziness and nausea.

Metheptazine is not listed as a controlled substance under the Controlled Substances Act 1970 in the United States.[2] The Canadian Controlled Drugs and Substances Act specifically excludes the phenazepine opioids from control.

References
  1. US Patent 2740777 PROCESS FOR THE PREPARATION OF HEXAHYDRO-1,3-DIMETHYL- 4-PHENYLAZEPINE-4-CARBOXYLIC ACID, ETHYL ESTER
  2. http://www.deadiversion.usdoj.gov/quotas/conv_factor/index.html


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